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产品介绍
产品介绍
产品信息
抗原名称
D4.4 receptor,D4.2 receptor,D4.7 receptor
商品描述
A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM).
分子量
320.43
纯度
98%
可溶性
DMSO : 51.67 mg/mL (161.25 mM; Need ultrasonic)
In vitro(体外研究)
A-381393 exhibits weak affinity at 5-HT1A, Sigma 2, Adenoceptor α1A, Adenoceptor α2C, Histamine H1, with Kis of 1365, 8600, 2044, 1912 and 2962 nM, respectively.
背景
分子式
C20H24N4
CAS号
726174-00-1
制备和贮存
保存方式
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
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