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GSK2801
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产品介绍
产品介绍
产品信息
抗原名称
BAZ2B ,BAZ2A
商品描述
GSK2801 is a very potent inhibitor of the BAZ2 family of bromodomain containing proteins.
分子量
371.45
纯度
>98%
可溶性
DMSO 74 mg/mL warmed (199.21 mM)
Ethanol 7 mg/mL warmed (18.84 mM)
Ethanol 7 mg/mL warmed (18.84 mM)
外观
Powder
In vitro(体外研究)
In U2OS cells transfected with mutant BAZ2A (N1873F), GSK2801 (1 μM) accelerates FRAP half-recovery time by displacing BAZ2A from chromatin.
In vivo(体内研究)
In male CD1 mice, GSK2801 (30 mg/kg, p.o. and i.p.) has reasonable in vivo exposure after oral dosing, modest clearance, and reasonable plasma stability.
背景
别名
GSK-2801, GSK 280
分子式
C20H21NO4S
CAS号
1619994-68-1
制备和贮存
保存方式
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
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