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NVP-BKM120 Hydrochloride
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产品介绍
产品介绍
产品信息
商品描述
NVP-BKM120 Hydrochloride is a selective PI3K inhibitor of p110??/??/??/?? with IC50 of 52 nM/166 nM/116 nM/262 nM, respectively. Reduced potency against VPS34, mTOR, DNAPK, with little activity to PI4K??.

分子量
446.85

纯度
>98%

可溶性
10 mM in DMSO

背景
别名
BKM-120 hydrochloride, BKM120 hydrochloride, BKM 120 hydrochloride

分子式
C18H21F3N6O2.HCl

CAS号
1312445-63-8

制备和贮存
保存方式
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
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