RX 821002 hydrochloride (10 mg)

11957683

Potent, selective α_2D antagonist

270.72

2-(2,3-Dihydro-2-methoxy-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole hydrochloride

Potent, selective α₂-adrenoceptor antagonist with very low affinity for imidazoline sites. Displays selectivity for the α_2D over the α_2A subtypes (pK_d values are 9.7 and 8.2 respectively).

≥99% (HPLC)

Soluble to 100 mM in water and to 100 mM in DMSO

Cl.COC1(COC2=CC=CC=C2O1)C1=NCCN1

C₁₂H₁₄N₂O₃.HCl

109544-45-8