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产品介绍
产品介绍
产品信息
商品描述
Xli 093 is an α5 subtype selective benzodiazepine/GABAA receptor antagonist. Xli 093 shows Ki = 5 nM at the α5 receptor in Ltk- cell membranes expressing human α5β3γ2 receptors; little or no affinity at other BDZ/ GABAA subtypes; does not trigger chloride currents in any subtype of tested subtypes, up to 1 μM in concentration; dose-dependently and completely inhibits diazepam stimulated currents in α5β3γ2 receptors.
分子量
602.60
可溶性
Soluble in DMSO: ~16 mg/mL: water: insoluble
外观
Powder
应用
实验应用
Α5 subtype selective benzodiazepine/GABAA receptor antagonist
背景
别名
Bis[8-ethynyl-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic acid] 1,3-propanediyl ester
分子式
C33H26N6O6
CAS号
646066-59-3(anhydrous)
制备和贮存
保存方式
Store at 4° C
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